OnCo
pathwaysPathway

Chromosomal instability & aneuploidy

Most cancers have the wrong number of chromosomes and keep shuffling them at every division. This chaos fuels evolution and drug resistance, but it also stresses the cell and can trigger immune alarms, a double edge that researchers are trying to exploit.

Chromosomal instability (CIN) arises from mitotic errors, whole-genome doubling, replication stress, and centrosome amplification; it produces aneuploidy, micronuclei, chromothripsis, and ecDNA (extrachromosomal oncogene amplicons). Consequences: intratumour heterogeneity and rapid adaptation (TRACERx), cytosolic DNA that activates cGAS-STING (immunogenic in bursts, tolerated chronically via non-canonical NF-κB), and proteotoxic and metabolic stress that creates dependencies (KIF18A, spindle assembly checkpoint, BCL-XL). CIN is a poor-prognosis marker across cancers; ecDNA drives resistance to targeted therapy in glioblastoma and others.

In one picture

Chromosomal instability is a library that reshuffles and duplicates random shelves every night. Most rearrangements are useless, some ruin the building, but occasionally one yields a book the librarian needs to survive a new rule, and the mess itself keeps the fire alarms twitching.

Diagram

top
Light up a product:+6 more via the Connected tab
Mitotic errors, WGDChromosomal instabilityAneuploidy / karyotype he…Micronuclei → cytosolic D…cGAS–STINGecDNA oncogene amplificat…Clonal evolution, resista…Dependencies: KIF18A, SAC…TP53 loss permitsactivatesinhibitsdruggable target (click)hit by selected productescape route

How drugs attack it

4top
  • KIF18A inhibitors (sovilnesib) selectively kill CIN-high cells; phase 1/2 in ovarian and TNBC
  • ecDNA-directed strategies (CHK1 inhibition, transcriptionreplication conflict) from the Cancer Grand Challenges eDyNAmiC team
  • STING pathway modulation; radiation exploits CIN
  • Aneuploidy scores (TRACERx) as prognostic biomarkers

Notes

top
  • Leading programmes: Swanton (Crick/UCL, TRACERx, CIN and immune evasion); Bakhoum (MSK, CIN–STING); Mischel (Stanford) and the eDyNAmiC Cancer Grand Challenge on ecDNA; Sheltzer (Yale) on aneuploidy dependencies.

Key papers

2top

Connected

20top

Pages like this

not linked directly; found by shared links