OnCo
drugsProductNot mapped hereapproved

Ensartinib

A Chinese-developed ALK pill approved in the US in December 2024 for first-line ALK-positive lung cancer.

eXalt3 (JAMA Oncol 2021): PFS 25.8 vs 12.7 months versus crizotinib in ALK-TKI-naive NSCLC. Approved in China 2020 (post-crizotinib), 2022 first line; US approval December 2024 (Xcovery). Rash is the characteristic toxicity.

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Ensartinib
PubChem
Modality
Small-molecule ALK TKI (second generation)
Mechanism
Potent ALK inhibitor with activity against crizotinib-resistant mutations and CNS penetration.
Brand / code
Ensacove
Medicare
Part D (self-administered)

Oral, self-administered, so it is a Part D drug: covered through a stand-alone Part D plan or Medicare Advantage drug benefit, usually on the specialty tier with 25 to 33% coinsurance until the annual cap ($2,000 in 2025, $2,100 in 2026). FDA-approved December 2024.

Commercial insurance
covered with prior authorisation

Covered for FDA-labelled and NCCN-listed uses, but almost always behind prior authorisation confirming diagnosis, biomarker and line of therapy; dispensed through a specialty pharmacy.

Part D out-of-pocket capped at $2,000 (2025) / $2,100 (2026). Medicare patients cannot use manufacturer co-pay cards; charity funds (PAN, HealthWell, CancerCare) and the Extra Help subsidy are the routes.

Sources: Medicare.gov: Drug coverage (Part D) · Medicare.gov: Costs for Medicare drug coverage (annual out-of-pocket cap). Not medical or financial advice; verify with your plan.

Not appraisedSearch NICE
Notes
No UK marketing authorisation as of September 2026, so no NICE appraisal. Access only through a clinical trial or a company early access scheme.
NHS England
Not routinely funded

Sources: NICE search: ensartinib. Funding decisions are indication-specific and change monthly; verify with NICE and your treating team.

Regulatory

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Approvals

RegionYearIndication
CN2020ALK-positive NSCLC after crizotinib
US2024ALK-positive locally advanced or metastatic NSCLC, ALK-inhibitor-naive

Trials

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Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
Ensartinib
intervention: Ensartinib
Open on ClinicalTrials.gov →

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Latest papers

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Latest papers · live from Europe PMC
Open in Europe PMC

Query for this drug: (TITLE:"Ensartinib" OR ABSTRACT:"Ensartinib" OR TITLE:"Ensacove" OR ABSTRACT:"Ensacove") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about Ensartinib, not a curated reading list.

Connected

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