OnCo
drugsProductNot mapped hereapproved

5-Aminolevulinic acid (oral, for glioma surgery)

A drink taken before brain surgery that makes high-grade glioma glow under blue light, letting surgeons remove more tumour safely.

Stummer randomised trial (Lancet Oncol 2006): complete resection 65% vs 36% and better 6-month PFS. EMA approved 2007; FDA 2017 (first optical imaging agent for brain surgery). Also used topically for actinic keratosis photodynamic therapy (Levulan/Ameluz) and in bladder (hexaminolevulinate).

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5-Aminolevulinic acid
PubChem
Modality
Fluorescence-guided surgery agent (protoporphyrin IX precursor)
Mechanism
Oral 5-ALA is taken up by glioma cells and converted to protoporphyrin IX, which fluoresces pink-red under blue light (400-410 nm) through the surgical microscope.
Brand / code
Gleolan / Gliolan
Medicare
Part B (clinician-administered)

Oral solution given two to four hours before glioma surgery in the hospital, so it is a surgical supply bundled into the Part A inpatient stay rather than a pharmacy benefit.

Commercial insurance
covered on label

Bundled into the craniotomy claim; no separate authorisation is typical.

Sources: Medicare.gov: Chemotherapy · Medicare.gov: Prescription drugs (outpatient, Part B) · Medicare.gov: Inpatient hospital care (Part A). Not medical or financial advice; verify with your plan.

NICE recommendedSearch NICE
Appraised for
Fluorescence-guided resection of high-grade glioma
Notes
Recommended in NICE guideline NG99 (brain tumours, 2018) rather than a TA; routinely used in NHS neurosurgical centres.
NHS England
Routinely funded for the appraised indication (or via managed access)

Sources: NICE search: 5-aminolevulinic acid (Gliolan). Funding decisions are indication-specific and change monthly; verify with NICE and your treating team.

Regulatory

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Approvals

RegionYearIndication
EU2007Visualisation of malignant tissue during surgery for WHO grade III-IV glioma
US2017Imaging agent for visualisation of malignant tissue during glioma surgery (suspected high-grade)

Trials

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Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
5-Aminolevulinic acid (oral, for glioma surgery)
intervention: 5-Aminolevulinic acid
Open on ClinicalTrials.gov →

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Latest papers

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Latest papers · live from Europe PMC
Open in Europe PMC

Query for this drug: (TITLE:"5-Aminolevulinic acid" OR ABSTRACT:"5-Aminolevulinic acid" OR TITLE:"oral, for glioma surgery" OR ABSTRACT:"oral, for glioma surgery" OR TITLE:"Gleolan" OR ABSTRACT:"Gleolan" OR TITLE:"Gliolan" OR ABSTRACT:"Gliolan") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about 5-Aminolevulinic acid (oral, for glioma surgery), not a curated reading list.

Connected

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